Numero ya cas: 168273-06-1 Imiterere ya molekulari ： C22H21Cl3N4O
| Ingingo yo gushonga | 154.7 ° C. |
| Ubucucike | 1.299 |
| ububiko bwa temp | nta mbogamizi. |
| gukemura | Gukemura muri DMSO (kugeza kuri mg / ml 20) cyangwa muri Ethanol (kugeza kuri mg / ml 20).dimethyl sulfoxide no kudashonga muri benzene cyangwa hexane. |
| ibikorwa byiza | N / A. |
| Kugaragara | cyera kugeza cyoroshye umuhondo wa kirisiti |
| Isuku | ≥98% |
ni anti-antagonist ya reseptor ya urumogi (CB1).Ikora muguhitamo guhitamo reseptor ya CB1 iboneka mubwonko no mubice bya periferique bifite akamaro kanini muri glucose na lipide metabolism, harimo tipusi ya adipose, umwijima, inzira ya gastrointestinal, n'imitsi.Rero, bigize uburyo bwo kuvura umubyibuho ukabije hamwe nimpamvu zitera umutima.Nkumuti wa anorectic antiobesity, wakoreshejwe nkumugereka wimirire nimyitozo ngororamubiri kubarwayi bafite umubyibuho ukabije cyangwa ufite ibiro byinshi bafite ingaruka ziterwa n’uburayi mu 2006. Nubwo bimeze bityo ariko, havuzwe ingaruka mbi zirimo kwiyahura, kwiheba, no guhangayika, zishingiye kuri rimonadant. ku isi hose mu 2008.
Urumogi rwa Andogène rufitanye isano n'ingaruka zishimishije za nikotine, nk'urumogi rwakira urumogi, narwo rurageragezwa nk'umuti ushobora kurwanya itabi.
ni immunomodulatory CB1 reseptor inverse agonist
Baza Muganga inama mbere
